X-Nico

unusual facts about partial agonist



OSU-6162

OSU-6162 (PNU-96391) is a compound which acts as a partial agonist at both 2A5-HT2A receptors.

Α5IA

It binds to the partial agonist effect at α2 likely to be responsible for the lack of anxiety produced by this drug when compared to older α5-preferring inverse agonists such as L-655,708.


see also

C20H26N2O4

Binospirone, a partial agonist at 5HT1A somatodendritic autoreceptors